human Adrenergic α2C receptor is also available for Aequorin (calcium), GTPγS and radioligand binding competition assays

Target Information

Family :
Adrenergic
Receptor :

α2C

Species :
Homo sapiens
Accession number :
NP_000674.2

Assay Information

Cat. Number :
ES-032C
Method :
HTRF
Assay Type :
cAMP – Gi mode
Source :
CHO-K1

Testing Information

Mode:
agonist
Reference agonist:
UK 14,304
EC50:
12.5nM*
#ALT#

Mode:
antagonist
Reference antagonist:
ARC 239
IC50:
688nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot