Safety panel

Profile your compounds against a panel of 44 GPCR, ion channel, transporters and enzymes for potential safety issues.


Family Target Readout Family Target Readout
Adenosine A2A Binding Histamine H2 Binding
Adrenergic α1a Binding Melatonin MT1 Binding
α2a Binding MT2 Binding
β2 Binding Muscarinic Non selective Binding
Cannabinoid CB1 Binding Serotonin 5-HT1A Binding
Dopamine D1 Binding 5-HT1B Binding
D2S Binding 5-HT2A Binding
Opioid σ Binding 5-HT2B Binding
δ Binding Cholecystokinin CCK1 Binding
κ Binding Endothelin ETA Binding
μ Binding ETB Binding
Histamine H1 Binding Vasopressin V1a Binding


Family Target Readout
Amine transporter DAT Binding
NET Binding
SERT Binding

Ion channels

Family Target Readout
Ca2+ channel L-type, DHP site Binding
L-type, Verapamil site Binding
K+ channel hERG Binding
Serotonin 5-HT3 Binding
GABA BZD (Central) Binding
NMDA GRIN1 Binding
Nicotinic α4β2 Binding


Family Target Readout
Acetylcholinesterase AChE Fluorescence
Cyclooxygenase COX-2 Colorimetric
Monoamine Oxidase MAO-A Luminescence
Phosphodiesterase PDE-3 HTRF
Phosphodiesterase PDE-4 HTRF
Cytochrome P450 CYP1A2 Luminescence
CYP2C9 Luminescence
CYP2D6 Luminescence
CYP2E1 Luminescence
CYP3A4 Luminescence

Custom profile

If you don’t find a profiling that suits your needs, don’t hesitate to contact us and let us know what you are looking for. We’ll be happy to help you out and design a tailor-made panel!

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