human Ghrelin receptor (GHSR) is also validated for Aequorin (calcium) and radioligand binding competition assays

Target Information

Family :
Ghrelin
Receptor :

GHSR

Species :
Homo sapiens
Accession number :
NP_940799.1

Assay Information

Cat. Number :
FAST-0135I
Method :
HTRF
Assay Type :
IPOne
Source :
CHO-K1

Testing Information

Mode:
agonist
Reference agonist:
Ghrelin
EC50:
1.83nM*
#ALT#

Mode:
antagonist
Reference antagonist:
[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P
IC50:
382nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot