FAST-0903C
Orphan GPR17 cAMP
human GPR17 receptor is also validated for Aequorin (calcium) and IPOne assays
Target Information
- Family :
- Orphan
- Receptor :
-
GPR17
- Species :
- Homo sapiens
- Accession number :
- NP_001154888.1
Assay Information
- Cat. Number :
- FAST-0903C
- Method :
- HTRF
- Assay Type :
- cAMP – Gi mode
- Source :
- CHO-K1
Testing Information
- Mode:
- agonist
- Reference agonist:
- MDL 29,951
- EC50:
- 6.01nM*
- Mode:
- antagonist
- Reference antagonist:
- HAMI3379
- IC50:
- 372nM*
- Standard TAT :
- 15 Business Days
- Fast TAT :
- 5 Business Days
- * Value is subjected to variation from lot to lot