FAST-040G
Cannabinoid CB1 GTPγS
human Cannabinoid CB1 receptor is also available for cAMP, ERK1/2 and radioligand binding competition assays
Target Information
- Family :
- Cannabinoid
- Receptor :
-
CB1
- Species :
- Homo sapiens
- Accession number :
- NP_057167.2
Assay Information
- Cat. Number :
- FAST-040G
- Method :
- SPA
- Assay Type :
- GTPγS
- Source :
- CHO-K1
Testing Information
- Mode:
- agonist
- Reference agonist:
- CP 55,940
- EC50:
- 17.3nM*
- Mode:
- antagonist
- Reference antagonist:
- AM 251
- IC50:
- 13.3nM*
- Mode:
- inverse agonist
- Reference inverse agonist:
- AM 251
- IC50:
- 1.75nM*
- Standard TAT :
- 15 Business Days
- Fast TAT :
- 5 Business Days
- * Value is subjected to variation from lot to lot