FAST-0440C
Protease-activated PAR2 cAMP
human Proteinase-activated receptor PAR2 is also validated for Aequorin (calcium), IPOne and GTPγS assays
Target Information
- Family :
- Protease-activated
- Receptor :
-
PAR2
- Species :
- Homo sapiens
- Accession number :
- NP_005233.3
Assay Information
- Cat. Number :
- FAST-0440C
- Method :
- HTRF
- Assay Type :
- cAMP – Gi mode
- Source :
- CHO-K1-mt aequorin
Testing Information
- Mode:
- agonist
- Reference agonist:
- SLIGRL-NH2
- EC50:
- 1.6µnM*
- Mode:
- Antagonist
- Reference antagonist:
- AZ3451
- IC50:
- 14.0nM*
- Standard TAT :
- 15 Business Days
- Fast TAT :
- 5 Business Days
- * Value is subjected to variation from lot to lot