human Adenosine A2A receptor is also available for cAMP, GTPγS and radioligand binding competition assays

Target Information

Family :
Adenosine
Receptor :

A2A

Species :
Homo sapiens
Accession number :
NP_00666.2

Assay Information

Cat. Number :
FAST-002A
Method :
luminescence
Assay Type :
aequorin (calcium)
Source :
HEK293-mt aequorin-Gα16

Testing Information

Mode:
agonist
Reference agonist:
NECA
EC50:
103nM*
#ALT#

Mode:
antagonist
Reference antagonist:
ZM 241385
IC50:
1.36nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot