human Bombesin BB2 receptor is also available for radioligand binding competition assays

Target Information

Family :
Bombesin
Receptor :

BB2

Species :
Homo sapiens
Accession number :
NP_005305.1

Assay Information

Cat. Number :
FAST-023A
Method :
luminescence
Assay Type :
aequorin (calcium)
Source :
CHO-K1-mt aequorin-Gα16

Testing Information

Mode:
agonist
Reference agonist:
Gastrin-releasing peptide (GRP)
EC50:
35.9pM*
#ALT#

Mode:
antagonist
Reference antagonist:
[D-Phe12] Bombesin
IC50:
18.2nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot