human Cannabinoid CB1 receptor is also available for GTPγS, ERK1/2 and radioligand binding competition assays

Target Information

Family :
Cannabinoid
Receptor :

CB1

Species :
Homo sapiens
Accession number :
NP_057167.2

Assay Information

Cat. Number :
FAST-040C
Method :
HTRF
Assay Type :
cAMP – Gi mode
Source :
CHO-K1

Testing Information

Mode:
agonist
Reference agonist:
CP 55,940
EC50:
0.67nM*
#ALT#

Mode:
antagonist
Reference antagonist:
AM 251
IC50:
12.5nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot