human CXCR1 receptor is also validated for Aequorin (calcium), GTPγS and radioligand binding competition assays

Target Information

Family :
Chemokine
Receptor :

CXCR1

Species :
Homo sapiens
Accession number :
NP_000625.1

Assay Information

Cat. Number :
FAST-071C
Method :
HTRF
Assay Type :
cAMP – Gi mode
Source :
CHO-K1

Testing Information

Mode:
agonist
Reference agonist:
CXCL8 (IL-8)
EC50:
0.22nM*
#ALT#

Mode:
Antagonist
Reference antagonist:
SB265610
IC50:
275nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot