human CXCR4 receptor is also validated for Aequorin (calcium), GTPγS and radioligand binding competition assays

Target Information

Family :
Chemokine
Receptor :

CXCR4

Species :
Homo sapiens
Accession number :
NP_003458.1

Assay Information

Cat. Number :
FAST-077C
Method :
HTRF
Assay Type :
cAMP – Gi mode
Source :
CHO-K1

Testing Information

Mode:
agonist
Reference agonist:
CXCL12 (SDF-1α)
EC50:
1.08nM*
#ALT#

Mode:
antagonist
Reference antagonist:
AMD 3100
IC50:
961nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot