human CRF1 receptor is also validated for cAMP, GTPγS and radioligand binding competition assays

Target Information

Family :
Corticotropin-releasing factor
Receptor :

CRF1

Species :
Homo sapiens
Accession number :
NP_004373.2

Assay Information

Cat. Number :
FAST-095A
Method :
luminescence
Assay Type :
aequorin (calcium)
Source :
CHO-K1-mt aequorin-Gα16

Testing Information

Mode:
agonist
Reference agonist:
Urocortin
EC50:
29.6nM*
#ALT#

Mode:
antagonist
Reference antagonist:
CRF 9-41
IC50:
653nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot