human Endothelin ETA receptor is also validated for radioligand binding competition assays

Target Information

Family :
Endothelin
Receptor :

ETA

Species :
Homo sapiens
Accession number :
NP_001948.1

Assay Information

Cat. Number :
FAST-0105A
Method :
luminescence
Assay Type :
aequorin (calcium)
Source :
CHO-K1-mt aequorin

Testing Information

Mode:
agonist
Reference agonist:
Endothelin
EC50:
0.022nM*
#ALT#

Mode:
antagonist
Reference antagonist:
BQ 123
IC50:
1.56nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot