human GPR84 receptor is also validated for Aequorin (calcium), GTPγS, ERK1/2 and internalisation assays

Target Information

Family :
Free fatty acid
Receptor :

GPR84

Species :
Homo sapiens
Accession number :
NP_065103.1

Assay Information

Cat. Number :
FAST-0935C
Method :
HTRF
Assay Type :
cAMP – Gi mode
Source :
CHO-K1

Testing Information

Mode:
agonist
Reference agonist:
Capric acid
EC50:
23.6µM*
#ALT#
Mode:
agonist
Reference agonist:
Embelin
EC50:
44.9nM*
#ALT#
Mode:
antagonist
Reference antagonist:
GLPG1205
IC50:
14.1nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot