human GABA B1a/B2  heteromer is also validated for cAMP, GTPγS and radioligand binding competition assays

Target Information

Family :
GABA B
Target :
GABA B1a/B2
Species :
Homo sapiens
Accession number :
CAA09939.1 / CAA09942.1

Assay Information

Cat. Number :
FAST-0120A
Method :
luminescence
Assay Type :
aequorin (calcium)
Source :
CHO-K1-mt aequorin-Gα16

Testing Information

Mode:
agonist
Reference agonist:
GABA
EC50:
1.49µM*
#ALT#

Mode:
antagonist
Reference antagonist:
CGP 54626
IC50:
11.8nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot