FAST-0120G
GABA GABA B1a/B2 GTPγS
human GABA B1a/B2 heteromer is also validated for Aequorin (calcium), cAMP and radioligand binding competition assays
Target Information
- Family :
- GABA B
- Target :
- GABA B1a/B2
- Species :
- Homo sapiens
- Accession number :
- CAA09939.1 / CAA09942.1
Assay Information
- Cat. Number :
- FAST-0120G
- Method :
- SPA
- Assay Type :
- GTPγS
- Source :
- CHO-K1
- Mode:
- agonist
- Reference agonist:
- GABA
- Ec50:
- 11.2µM*
Testing Information
- Mode:
- agonist
- Reference agonist:
- SKF 97541
- EC50:
- 6.89µM*
- Mode:
- antagonist
- Reference antagonist:
- CGP 54626
- IC50:
- 21.8nM*
- Standard TAT :
- 15 Business Days
- Fast TAT :
- 5 Business Days
- * Value is subjected to variation from lot to lot