human GABA B1b/B2  heteromer is validated for cAMP assays

Target Information

Family :
GABA B
Target :
GABA B1b/B
Species :
Homo sapiens
Accession number :
CAA09940.1 / CAA09942.1

Assay Information

Cat. Number :
FAST-0122C
Method :
HTRF
Assay Type :
cAMP – Gi mode
Source :
CHO-K1

Testing Information

Mode:
agonist
Reference agonist:
GABA
EC50:
20.6nM*
#ALT#
Mode:
Antagonist
Reference antagonist:
CGP 54,626
IC50:
3.36nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot