human Glutamate mGlu1 receptor is also available for cAMP assays

Target Information

Family :
Glutamate
Receptor :

mGlu1

Species :
Homo sapiens
Accession number :
AAA87843.1

Assay Information

Cat. Number :
FAST-0152A
Method :
luminescence
Assay Type :
aequorin (calcium)
Source :
CHO-K1-mt aequorin (inducible)

Testing Information

Mode:
agonist
Reference agonist:
Glutamate
EC50:
1.2µM*
#ALT#

Mode:
antagonist
Reference antagonist:
JNJ 16259685
IC50:
8.88nM*
#ALT#
Mode:
PAM
Reference PAM:
CPPHA
EC50:
853nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot