human Glutamate mGlu4 receptor is also available for GTPγS assays

Target Information

Family :
Glutamate
Receptor :

mGlu4

Species :
Homo sapiens
Accession number :
NP_000832.1

Assay Information

Cat. Number :
FAST-0150C
Method :
HTRF
Assay Type :
cAMP – Gi mode
Source :
CHO-K1

Testing Information

Mode:
agonist
Reference agonist:
Glutamate
EC50:
3.8µM*
#ALT#

Mode:
antagonist
Reference antagonist:
LY 341495
IC50:
10.5µM*
#ALT#
Mode:
PAM
Reference PAM:
VU 0155041
EC50:
822nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot