FAST-0151A
Glutamate mGlu5 Aequorin
human Glutamate mGlu5 receptor is also validated for IPOne and radioligand binding competition assays
Target Information
- Family :
- Glutamate (metabotropic)
- Receptor :
-
mGlu5
- Species :
- Homo sapiens
- Accession number :
- NP_000833.1
Assay Information
- Cat. Number :
- FAST-0151A
- Method :
- luminescence
- Assay Type :
- aequorin (calcium)
- Source :
- CHO-K1-mt aequorin (inducible)
Testing Information
- Mode:
- agonist
- Reference agonist:
- Glutamate
- EC50:
- 581nM*
- Mode:
- antagonist
- Reference antagonist:
- MPEP
- IC50:
- 8.13nM*
- Mode:
- PAM
- Reference PAM:
- DFB
- EC50:
- 519nM*
- Standard TAT :
- 15 Business Days
- Fast TAT :
- 5 Business Days
- * Value is subjected to variation from lot to lot