human Glutamate mGlu5 receptor is also validated for Aequorin (calcium) and radioligand binding competition assays

Target Information

Family :
Glutamate (metabotropic)
Receptor :

mGlu5

Species :
Homo sapiens
Accession number :
NP_000833.1

Assay Information

Cat. Number :
FAST-0151I
Method :
HTRF
Assay Type :
IPOne
Source :
CHO-K1-mt aequorin (inducible)

Testing Information

Mode:
agonist
Reference agonist:
Glutamate
EC50:
418nM*
#ALT#

Mode:
antagonist
Reference antagonist:
MPEP
IC50:
284nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot