FAST-0172G
Histamine H3 GTPγS
human Histamine H3 receptor is also validated for Aequorin (calcium), cAMP and radioligand binding competition assays
Target Information
- Family :
- Histamine
- Receptor :
-
H3
- Species :
- Homo sapiens
- Accession number :
- NP_009163.2
Assay Information
- Cat. Number :
- FAST-0172G
- Method :
- SPA
- Assay Type :
- GTPγS
- Source :
- CHO-K1
Testing Information
- Mode:
- agonist
- Reference agonist:
- (R)-(-)-α-Methylhistamine
- EC50:
- 0.81nM*
- Mode:
- antagonist
- Reference antagonist:
- Clobenpropit
- IC50:
- 7.45nM*
- Standard TAT :
- 15 Business Days
- Fast TAT :
- 5 Business Days
- * Value is subjected to variation from lot to lot