human Histamine H4 receptor is also validated for GTPγS and radioligand binding competition assays

Target Information

Family :
Histamine
Receptor :

H4

Species :
Homo sapiens
Accession number :
NP_067637.2

Assay Information

Cat. Number :
FAST-0173A
Method :
luminescence
Assay Type :
aequorin (calcium)
Source :
CHO-K1-mt aequorin-Gα16

Testing Information

Mode:
agonist
Reference agonist:
Histamine
EC50:
649nM*
#ALT#

Mode:
antagonist
Reference antagonist:
Thioperamide
IC50:
224nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot