FAST-1306
Ion channel CaV1.2 (Verapamil) Binding
Radioligand binding competition assays for the Verapamil site of the Cav1.2 (L-type) voltage-gated calcium ion channel are available for testing
Target Information
- Family :
- Ion channel
- Target :
- Cav1.2 (L-type) (Varapamil site)
- Species :
- Rattus norvegicus
Assay Information
- Cat. Number :
- FAST-1306
- Method :
- radiometric
- Assay Type :
- filtration binding
- Source :
- rat brain membrane preparation
Testing Information
- Mode:
- competition
- Tracer:
- [N-methyl-3H] Desmethoxyverapamil
- Tracer concentration:
- 2nM
- Reference competitor:
- Methoxyverapamil
- IC50:
- 649nM*
- Standard TAT :
- 15 Business Days
- Fast TAT :
- 5 Business Days
- * Value is subjected to variation from lot to lot