human GPR55 receptor is also available for internalisation assay

Target Information

Family :
Lysophospholipid
Receptor :

GPR55

Species :
Homo sapiens
Accession number :
NP_005674.2

Assay Information

Cat. Number :
FAST-0922A
Method :
luminescence
Assay Type :
aequorin (calcium)
Source :
CHO-K1-mt aequorin-Gq13

Testing Information

Mode:
agonist
Reference agonist:
AM 251
EC50:
2.23µM*
#ALT#
Mode:
agonist
Reference agonist:
Lysophosphatidylinositol (LPI)
EC50:
11.6µM*
#ALT#
Mode:
antagonist
Reference antagonist:
ML 193
IC50:
975nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot