human MCH1 receptor is also validated for cAMP, GTPγS and radioligand binding competition assays

Target Information

Family :
Melanin-concentrating hormone
Receptor :

MCH1

Species :
Homo sapiens
Accession number :
NP_005288.3

Assay Information

Cat. Number :
FAST-0220A
Method :
luminescence
Assay Type :
aequorin (calcium)
Source :
CHO-K1-mt aequorin-Gα16

Testing Information

Mode:
agonist
Reference agonist:
MCH
EC50:
11.6nM*
#ALT#

Mode:
antagonist
Reference antagonist:
ATC 0175
IC50:
6.41nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot