FAST-0232C
Melanocortin MC3 cAMP
human Melanocortin MC3 receptor is also validated for radioligand binding competition assays
Target Information
- Family :
- Melanocortin
- Receptor :
-
MC3
- Species :
- Homo sapiens
- Accession number :
- AAC13541.1 I81V
Assay Information
- Cat. Number :
- FAST-0232C
- Method :
- HTRF
- Assay Type :
- cAMP – Gs mode
- Source :
- CHO-K1
Testing Information
- Mode:
- agonist
- Reference agonist:
- (Nle4,D-Phe7) α-MSH
- EC50:
- 0.29nM*
- Mode:
- antagonist
- Reference antagonist:
- SHU 9119
- IC50:
- 3.36nM*
- Standard TAT :
- 15 Business Days
- Fast TAT :
- 5 Business Days
- * Value is subjected to variation from lot to lot