human Melanocortin MC4 receptor is also validated for radioligand binding competition assays

Target Information

Family :
Melanocortin
Receptor :

MC4

Species :
Homo sapiens
Accession number :
NP_005903.2

Assay Information

Cat. Number :
FAST-0233C
Method :
HTRF
Assay Type :
cAMP – Gs mode
Source :
CHO-K1

Testing Information

Mode:
agonist
Reference agonist:
(Nle4,D-Phe7) α-MSH
EC50:
0.061nM*
#ALT#
Mode:
antagonist
Reference antagonist:
SHU 9119
IC50:
2.36nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot