FAST-0233C
Melanocortin MC4 cAMP
human Melanocortin MC4 receptor is also validated for radioligand binding competition assays
Target Information
- Family :
- Melanocortin
- Receptor :
-
MC4
- Species :
- Homo sapiens
- Accession number :
- NP_005903.2
Assay Information
- Cat. Number :
- FAST-0233C
- Method :
- HTRF
- Assay Type :
- cAMP – Gs mode
- Source :
- CHO-K1
Testing Information
- Mode:
- agonist
- Reference agonist:
- (Nle4,D-Phe7) α-MSH
- EC50:
- 0.061nM*
- Mode:
- antagonist
- Reference antagonist:
- SHU 9119
- IC50:
- 2.36nM*
- Standard TAT :
- 15 Business Days
- Fast TAT :
- 5 Business Days
- * Value is subjected to variation from lot to lot