FAST-0240A
Melatonin MT1 Aequorin
human Melatonin MT1 receptor is also validated for GTPγS and radioligand binding competition assays
Target Information
- Family :
- Melatonin
- Receptor :
-
MT1
- Species :
- Homo sapiens
- Accession number :
- NP_005949.1
Assay Information
- Cat. Number :
- FAST-0240A
- Method :
- luminescence
- Assay Type :
- aequorin (calcium)
- Source :
- CHO-K1-mt aequorin-Gα16
Testing Information
- Mode:
- agonist
- Reference agonist:
- 2-iodo-melatonin
- EC50:
- 6.63nM*
- Mode:
- antagonist
- Reference antagonist:
- Luzindole
- IC50:
- 1.42µM*
- Standard TAT :
- 15 Business Days
- Fast TAT :
- 5 Business Days
- * Value is subjected to variation from lot to lot