FAST-0260A
Muscarinic M1 Aequorin
human Muscarinic M1 receptor is also validated for IPOne, GTPgS and radioligand binding competition assays
Target Information
- Family :
- Muscarinic
- Receptor :
-
M1
- Species :
- Homo sapiens
- Accession number :
- NP_000729.2
Assay Information
- Cat. Number :
- FAST-0260A
- Method :
- luminescence
- Assay Type :
- aequorin (calcium)
- Source :
- CHO-K1-mt aequorin
Testing Information
- Mode:
- agonist
- Reference agonist:
- Acetylcholine
- EC50:
- 9.13nM*
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- Mode:
- antagonist
- Reference antagonist:
- 4-DAMP
- IC50:
- 0.59nM*
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- Standard TAT :
- 15 Business Days
- Fast TAT :
- 5 Business Days
- * Value is subjected to variation from lot to lot