human Muscarinic M1 receptor is also validated for Aequorin (calcium), IPOne and radioligand binding competition assays

Target Information

Family :
Muscarinic
Receptor :

M1

Species :
Homo sapiens
Accession number :
NP_000729.2

Assay Information

Cat. Number :
FAST-0260G
Method :
SPA
Assay Type :
GTPγS
Source :
CHO-K1

Testing Information

Mode:
agonist
Reference agonist:
Oxotremorine
EC50:
540nM*
#ALT#

Mode:
antagonist
Reference antagonist:
4-DAMP
IC50:
14.2nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot