human Muscarinic M3 receptor is also validated for Aequorin (calcium) and radioligand binding competition assays

Target Information

Family :
Muscarinic
Receptor :

M3

Species :
Homo sapiens
Accession number :
NP_000731.1

Assay Information

Cat. Number :
Es-212I
Method :
HTRF
Assay Type :
IPOne
Source :
CHO-K1

Testing Information

Mode:
agonist
Reference agonist:
Acetylcholine
EC50:
174nM*
#ALT#

Mode:
antagonist
Reference antagonist:
4-DAMP
IC50:
2.51nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot