ES-213A
Muscarinic M4 Aequorin
human Muscarinic M4 receptor is also validated for GTPγS and radioligand binding competition assays
Target Information
- Family :
- Muscarinic
- Receptor :
-
M4
- Species :
- Homo sapiens
- Accession number :
- NP_000732.1
Assay Information
- Cat. Number :
- ES-213A
- Method :
- luminescence
- Assay Type :
- aequorin (calcium)
- Source :
- CHO-K1-mt aequorin-Gα16
Testing Information
- Mode:
- agonist
- Reference agonist:
- Acetylcholine
- EC50:
- 63.1nM*
- Mode:
- antagonist
- Reference antagonist:
- N-Me-Scopolamine
- IC50:
- 0.068nM*
- Standard TAT :
- 15 Business Days
- Fast TAT :
- 5 Business Days
- * Value is subjected to variation from lot to lot