FAST-0379C
Opioid OP1 (delta) cAMP
human delta Opioid receptor, also known as OP1, is also validated for Aequorin (calcium), GTPγS and radioligand binding competition assays
Target Information
- Family :
- Opioid
- Receptor :
-
OP1
- Species :
- Homo sapiens
- Accession number :
- ACG60644.1
Assay Information
- Cat. Number :
- FAST-0379C
- Method :
- HTRF
- Assay Type :
- cAMP – Gi mode
- Source :
- CHO-K1
Testing Information
- Mode:
- agonist
- Reference agonist:
- SNC 80
- EC50:
- 17.1nM*
- Mode:
- antagonist
- Reference antagonist:
- Naltrindol
- IC50:
- 1.01nM*
- Mode:
- PAM
- Reference PAM:
- BMS 986187
- EC50:
- 165nM*
- Standard TAT :
- 15 Business Days
- Fast TAT :
- 5 Business Days
- * Value is subjected to variation from lot to lot