FAST-0379G
Opioid OP1 (delta) GTPγS
human delta Opioid receptor, also known as OP1, is also validated for Aequorin (calcium), cAMP and radioligand binding competition assays
Target Information
- Family :
- Opioid
- Receptor :
-
OP1
- Species :
- Homo sapiens
- Accession number :
- ACG60644.1
Assay Information
- Cat. Number :
- FAST-0379G
- Method :
- SPA
- Assay Type :
- GTPγS
- Source :
- CHO-K1
Testing Information
- Mode:
- agonist
- Reference agonist:
- SNC 80
- EC50:
- 3.44nM*
- Mode:
- antagonist
- Reference antagonist:
- Naltrindol
- IC50:
- 1.95nM*
- Mode:
- PAM
- Reference PAM:
- BMS 986187
- EC50:
- 4.63µM*
- Standard TAT :
- 15 Business Days
- Fast TAT :
- 5 Business Days
- * Value is subjected to variation from lot to lot