human kappa Opioid receptor, also known as OP2, is also validated for cAMP, GTPγS and radioligand binding competition assays

Target Information

Family :
Opioid
Receptor :

OP2

Species :
Homo sapiens
Accession number :
NP_000903.2

Assay Information

Cat. Number :
FAST-0380A
Method :
luminescence
Assay Type :
aequorin (calcium)
Source :
CHO-K1-mt aequorin

Testing Information

Mode:
agonist
Reference agonist:
GR 89696
EC50:
0.38nM*
#ALT#

Mode:
antagonist
Reference antagonist:
nor-Binaltorphimine
IC50:
1.28nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot