rat kappa Opioid receptor, also known as OP2, is validated for cAMP assays

Target Information

Family :
Opioid
Receptor :

OP2

Species :
Rattus norvegicus
Accession number :
NP_058863.1

Assay Information

Cat. Number :
FAST-0376C
Method :
HTRF
Assay Type :
cAMP – Gi mode
Source :
CHO-K1

Testing Information

Mode:
agonist
Reference agonist:
U-50488
EC50:
0.55nM*
#ALT#
Mode:
agonist
Reference agonist:
Nalfurafine
EC50:
7.75pM*
#ALT#
Mode:
antagonist
Reference antagonist:
nor-binaltorphimine
IC50:
0.47nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot