human kappa Opioid receptor, also known as OP2, is also validated for Aequorin (calcium), GTPγS and radioligand binding competition assays

Target Information

Family :
Opioid
Receptor :

OP2

Species :
Homo sapiens
Accession number :
NP_000903.2

Assay Information

Cat. Number :
FAST-0380C
Method :
HTRF
Assay Type :
cAMP – Gi mode
Source :
CHO-K1

Testing Information

Mode:
agonist
Reference agonist:
U-50488
EC50:
17.1nM*
#ALT#

Mode:
antagonist
Reference antagonist:
nor-Binaltorphimine
IC50:
0.46nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot