rat Orexin OX1 receptor is also validated for Aequorin (calcium) assays

Target Information

Family :
Orexin
Receptor :

OX1

Species :
Rattus norvegicus
Accession number :
NP_037196.1

Assay Information

Cat. Number :
FAST-0392I
Method :
HTRF
Assay Type :
IPOne
Source :
CHO-K1

Testing Information

Mode:
agonist
Reference agonist:
Orexin A
EC50:
2.92nM*
#ALT#
Mode:
antagonist
Reference antagonist:
SB 334867
IC50:
69.6nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot