human GPR17 receptor, short isoform, is also validated for cAMP and IPOne assays

Target Information

Family :
Orphan
Receptor :

GPR17

Species :
Homo sapiens
Accession number :
NP_001154888.1

Assay Information

Cat. Number :
FAST-0903A
Method :
luminescence
Assay Type :
aequorin (calcium)
Source :
CHO-K1-mt aequorin

Testing Information

Mode:
agonist
Reference agonist:
MDL 29,951
EC50:
360nM*
#ALT#

Mode:
antagonist
Reference antagonist:
HAMI3379
IC50:
1.61µM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot