mouse GPR17 receptor is also available for Aequorin (calcium) and IPOne assays

Target Information

Family :
Orphan
Receptor :

GPR17

Species :
Mus musculus
Accession number :
NP_001020552.1

Assay Information

Cat. Number :
FAST-0997C
Method :
HTRF
Assay Type :
cAMP – Gi mode
Source :
CHO-K1-mt aequorin

Testing Information

Mode:
agonist
Reference agonist:
MDL 29,951
EC50:
95.7.3nM*
#ALT#

Mode:
antagonist
Reference antagonist:
HAMI3379
IC50:
1.9µM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot