human GPR17 receptor, long isoform, is also validated for cAMP and IPOne assays

Target Information

Family :
Orphan
Species :
Homo sapiens
Accession number :
NP_005282.1

Assay Information

Cat. Number :
FAST-0996A
Method :
Luminescence
Assay Type :
aequorin (calcium)
Source :
CHO-K1-mt aequorin

Testing Information

Mode:
agonist
Reference agonist:
MDL 29,951
EC50:
980nM*
#ALT#

Mode:
Antagonist
Reference antagonist:
HAMI3379
IC50:
347nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot