FAST-0996G
Orphan GPR17-long GTPγS
human GPR17 receptor, long isoform, is also validated for Aequorin (calcium), cAMP and IPOne assays
Target Information
- Family :
- Orphan
- Receptor :
-
GPR17 long isoform
- Species :
- Homo sapiens
- Accession number :
- NP_005282.1
Assay Information
- Cat. Number :
- FAST-0996G
- Method :
- SPA
- Assay Type :
- GTPγS
- Source :
- CHO-K1-mt aequorin
Testing Information
- Mode:
- agonist
- Reference agonist:
- MDL 29,951
- EC50:
- 2.91µM*
- Mode:
- Antagonist
- Reference antagonist:
- HAMI3379
- IC50:
- 10.7µM*
- Standard TAT :
- 15 Business Days
- Fast TAT :
- 5 Business Days
- * Value is subjected to variation from lot to lot