rat GPR4 receptor is validated for cAMP assays

Target Information

Family :
pH sensing
Receptor :

GPR4

Species :
Rattus norvegicus
Accession number :
NP_001020851.1

Assay Information

Cat. Number :
FAST-0884C
Method :
HTRF
Assay Type :
cAMP – Gs mode
Source :
1321N1

Testing Information

Mode:
agonist
Reference agonist:
pH (H+)
EC50:
pH 7.4*
#ALT#

Mode:
antagonist
Reference antagonist:
NE 52-QQ57
IC50:
877nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot