human GPR68 receptor, also known as OGR1 for ovarian cancer G protein-coupled receptor 1, is validated for cAMP and IPOne assays

Target Information

Family :
pH sensing
Receptor :

GPR68

Species :
Homo sapiens
Accession number :
NP_003476.3

Assay Information

Cat. Number :
FAST-0928C
Method :
HTRF
Assay Type :
cAMP – Gs mode
Source :
1321N1

Testing Information

Mode:
agonist
Reference agonist:
pH (H+)
EC50:
pH 7.1*
#ALT#

Mode:
agonist
Reference agonist:
Ogerin
EC50:
996nM*
#ALT#
Mode:
antagonist
Reference antagonist:
Ogremorphin
IC50:
2.4µM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot