FAST-0439C
Protease-activated PAR1 cAMP
human Proteinase-activated receptor PAR1 is also validated for Aequorin (calcium), IPOne and GTPγS assays
Target Information
- Family :
- Protease-activated
- Receptor :
-
PAR1
- Species :
- Homo sapiens
- Accession number :
- NP_001983.2
Assay Information
- Cat. Number :
- FAST-0439C
- Method :
- HTRF
- Assay Type :
- cAMP – Gi mode
- Source :
- CHO-K1-mt aequorin
Testing Information
- Mode:
- agonist
- Reference agonist:
- TRAP-6
- EC50:
- 335nM*
- Mode:
- antagonist
- Reference antagonist:
- Vorapaxar
- IC50:
- 189nM*
- Standard TAT :
- 15 Business Days
- Fast TAT :
- 5 Business Days
- * Value is subjected to variation from lot to lot