human Proteinase-activated receptor PAR2 is also validated for Aequorin (calcium) and GTPγS assays

Target Information

Family :
Protease-activated
Receptor :

PAR2

Species :
Homo sapiens
Accession number :
NP_005233.3

Assay Information

Cat. Number :
FAST-0440I
Method :
HTRF
Assay Type :
IPOne
Source :
CHO-K1-mt aequorin

Testing Information

Mode:
agonist
Reference agonist:
Trypsin
EC50:
19.6nM*
#ALT#
Mode:
Antagonist
Reference antagonist:
AZ3451
IC50:
1.8µM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot