human Serotonin 5-HT3 channel is also available for radioligand binding competition assays

Target Information

Family :
Ion channel
Target :

5-HT3

Species :
Homo sapiens
Accession number :
NP_000860.3

Assay Information

Cat. Number :
FAST-0512A
Method :
luminescence
Assay Type :
aequorin (calcium)
Source :
HEK293-mt aequorin

Testing Information

Mode:
agonist
Reference agonist:
5-HT
EC50:
1.1µM*
#ALT#

Mode:
antagonist
Reference antagonist:
MDL 72222
IC50:
0.49nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot