rat Serotonin 5-HT4e receptor is validated for cAMP assays

Target Information

Family :
Serotonin
Receptor :

5-HT4e

Species :
Rattus norvegicus
Accession number :
NP_036985.1

Assay Information

Cat. Number :
FAST-0495C
Method :
HTRF
Assay Type :
cAMP – Gs mode
Source :
CHO-K1 (inducible)

Testing Information

Mode:
agonist
Reference agonist:
5-HT
EC50:
20.6
#ALT#

Mode:
antagonist
Reference antagonist:
GR 113808
IC50:
0.55nM*
#ALT#
Standard TAT :
15 Business Days
Fast TAT :
5 Business Days
* Value is subjected to variation from lot to lot