FAST-0553A
Vasopressin V1B Aequorin
rat Vasopressin V1B receptor are also validated for IPOne and radioligand binding competition assays
Target Information
- Family :
- Vasopressin
- Receptor :
-
V1B
- Species :
- Rattus norvegicus
- Accession number :
- BAA08242.1
Assay Information
- Cat. Number :
- FAST-0553A
- Method :
- luminescence
- Assay Type :
- Aequorin (calcium)
- Source :
- CHO-K1-mt-aequorin
Testing Information
- Mode:
- agonist
- Reference agonist:
- [Arg8]-Vasopressin
- EC50:
- 1.02nM*
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- Mode:
- antagonist
- Reference antagonist:
- SR 49059
- IC50:
- 334nM
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- Standard TAT :
- 15 Business Days
- Fast TAT :
- 5 Business Days
- * Value is subjected to variation from lot to lot